Knowledge (XXG)

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180: 165: 210: 195: 45: 120: 135: 60: 75: 105: 90: 225: 150: 30: 179: 164: 209: 194: 44: 119: 134: 59: 74: 104: 89: 224: 149: 29: 188:: NOVEL, POTENT SMALL MOLECULE INHIBITORS OF THE MOLECULAR CHAPERONE HSP90 DISCOVERED THROUGH STRUCTURE-BASED DESIGN 173:: NOVEL, POTENT SMALL MOLECULE INHIBITORS OF THE MOLECULAR CHAPERONE HSP90 DISCOVERED THROUGH STRUCTURE-BASED DESIGN 218:: 3-(5-CHLORO-2,4-DIHYDROXYPHENYL)-PYRAZOLE-4-CARBOXAMIDES AS INHIBITORS OF THE HSP90 MOLECULAR CHAPERONE 203:: 3-(5-CHLORO-2,4-DIHYDROXYPHENYL)-PYRAZOLE-4-CARBOXAMIDES AS INHIBITORS OF THE HSP90 MOLECULAR CHAPERONE 17: 53:: Human Hsp90 in complex with 17-desmethoxy-17-N,N-Dimethylaminoethylamino-Geldanamycin 68:: HUMAN HSP90-BETA WITH PU3 (9-BUTYL-8(3,4,5-TRIMETHOXY-BENZYL)-9H-PURIN-6-YLAMINE) 83:: Crystal Structures of human HSP90alpha complexed with dihydroxyphenylpyrazoles 113:: Crystal structure of human HSP90alpha complexed with dihydroxyphenylpyrazoles 98:: Crystal Structure of human HSP90alpha complexed with dihydroxyphenylpyrazoles 128:: HUMAN HSP90 GELDANAMYCIN-BINDING DOMAIN, ""CLOSED"" CONFORMATION 143:: HUMAN HSP90 GELDANAMYCIN-BINDING DOMAIN, ""OPEN"" CONFORMATION 233:: STRUCTURE-BASED DISCOVERY OF A NEW CLASS OF HSP90 INHIBITORS 158:: GELDANAMYCIN BOUND TO THE HSP90 GELDANAMYCIN-BINDING DOMAIN 8: 38:: HSP90 N-TERMINAL DOMAIN BOUND TO ADP-MG 25: 7: 24: 223: 208: 193: 178: 163: 148: 133: 118: 103: 88: 73: 58: 43: 28: 1: 249: 18:Template:PDB Gallery 240: 227: 212: 197: 182: 167: 152: 137: 122: 107: 92: 77: 62: 47: 32: 248: 247: 243: 242: 241: 239: 238: 237: 234: 228: 219: 213: 204: 198: 189: 183: 174: 168: 159: 153: 144: 138: 129: 123: 114: 108: 99: 93: 84: 78: 69: 63: 54: 48: 39: 33: 22: 21: 20: 12: 11: 5: 246: 244: 236: 235: 229: 222: 220: 214: 207: 205: 199: 192: 190: 184: 177: 175: 169: 162: 160: 154: 147: 145: 139: 132: 130: 124: 117: 115: 109: 102: 100: 94: 87: 85: 79: 72: 70: 64: 57: 55: 49: 42: 40: 34: 27: 23: 15: 14: 13: 10: 9: 6: 4: 3: 2: 245: 232: 226: 221: 217: 211: 206: 202: 196: 191: 187: 181: 176: 172: 166: 161: 157: 151: 146: 142: 136: 131: 127: 121: 116: 112: 106: 101: 97: 91: 86: 82: 76: 71: 67: 61: 56: 52: 46: 41: 37: 31: 26: 19: 230: 215: 200: 185: 170: 155: 140: 125: 110: 95: 80: 65: 50: 35: 16:< 231:2bz5 216:2byi 201:2byh 186:2bt0 171:2bsm 156:1yet 141:1yes 126:1yer 111:1yc4 96:1yc3 81:1yc1 66:1uym 51:1osf 36:1byq

Index

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1byq: HSP90 N-TERMINAL DOMAIN BOUND TO ADP-MG
1osf: Human Hsp90 in complex with 17-desmethoxy-17-N,N-Dimethylaminoethylamino-Geldanamycin
1uym: HUMAN HSP90-BETA WITH PU3 (9-BUTYL-8(3,4,5-TRIMETHOXY-BENZYL)-9H-PURIN-6-YLAMINE)
1yc1: Crystal Structures of human HSP90alpha complexed with dihydroxyphenylpyrazoles
1yc3: Crystal Structure of human HSP90alpha complexed with dihydroxyphenylpyrazoles
1yc4: Crystal structure of human HSP90alpha complexed with dihydroxyphenylpyrazoles
1yer: HUMAN HSP90 GELDANAMYCIN-BINDING DOMAIN, ""CLOSED"" CONFORMATION
1yes: HUMAN HSP90 GELDANAMYCIN-BINDING DOMAIN, ""OPEN"" CONFORMATION
1yet: GELDANAMYCIN BOUND TO THE HSP90 GELDANAMYCIN-BINDING DOMAIN
2bsm: NOVEL, POTENT SMALL MOLECULE INHIBITORS OF THE MOLECULAR CHAPERONE HSP90 DISCOVERED THROUGH STRUCTURE-BASED DESIGN
2bt0: NOVEL, POTENT SMALL MOLECULE INHIBITORS OF THE MOLECULAR CHAPERONE HSP90 DISCOVERED THROUGH STRUCTURE-BASED DESIGN
2byh: 3-(5-CHLORO-2,4-DIHYDROXYPHENYL)-PYRAZOLE-4-CARBOXAMIDES AS INHIBITORS OF THE HSP90 MOLECULAR CHAPERONE
2byi: 3-(5-CHLORO-2,4-DIHYDROXYPHENYL)-PYRAZOLE-4-CARBOXAMIDES AS INHIBITORS OF THE HSP90 MOLECULAR CHAPERONE
2bz5: STRUCTURE-BASED DISCOVERY OF A NEW CLASS OF HSP90 INHIBITORS

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