Knowledge (XXG)

Cantuzumab ravtansine

Source 📝

1329: 29: 87: 186: 1370: 347: 43: 756: 1389: 1363: 1288: 957: 313: 1177: 340: 1409: 814: 741: 646: 1404: 1356: 671: 268: 333: 1399: 656: 301: 761: 620: 144: 1305: 399: 864: 264: 1293: 1260: 1201: 1152: 1067: 691: 207: 1231: 1221: 1191: 982: 927: 854: 844: 721: 1206: 1195: 1157: 1047: 1032: 962: 937: 716: 470: 238: 226: 1057: 917: 686: 651: 306:
Antibody-Drug Conjugates and Immunotoxins: From Pre-Clinical Development to Therapeutic Applications
1394: 1336: 1172: 1142: 1137: 1122: 952: 799: 751: 711: 356: 211: 108: 53: 36: 410: 894: 445: 405: 269:"International Nonproprietary Names for Pharmaceutical Substances (INN). Proposed INN: List 105" 781: 600: 309: 1340: 117: 153: 218: 283: 1299: 1265: 932: 20: 1383: 1147: 1002: 555: 390: 1162: 1127: 1112: 1107: 1102: 1097: 1072: 1027: 1022: 1017: 1012: 997: 884: 859: 839: 701: 666: 605: 585: 395: 380: 325: 1270: 1244: 1239: 1211: 1187: 1182: 1117: 1092: 1082: 1052: 1042: 1007: 992: 977: 967: 947: 922: 907: 879: 829: 824: 819: 804: 794: 771: 766: 736: 681: 625: 615: 590: 580: 575: 570: 545: 520: 510: 505: 500: 490: 475: 460: 455: 440: 435: 425: 420: 415: 385: 1328: 1216: 1167: 1132: 1062: 1037: 987: 972: 912: 902: 874: 849: 789: 731: 726: 661: 641: 595: 565: 560: 550: 540: 535: 525: 515: 485: 480: 450: 430: 128: 28: 1087: 1077: 869: 834: 809: 746: 706: 696: 676: 610: 530: 495: 465: 243: 222: 58: 365: 70: 173: 302:"Linker technology and impact of linker design on ADC properties." 62: 164: 75: 329: 1344: 300:
Goldmacher VS, Singh R, Chittenden T, Kovtun Y (2013).
193: 210:
designed for the treatment of cancers. The humanized
1253: 1230: 893: 780: 634: 373: 364: 163: 143: 127: 107: 102: 86: 81: 69: 52: 42: 35: 116: 308:. New York: Springer. pp. 117–135 (131). 1364: 341: 8: 221:, ravtansine (DM4). It uses a more hindered 19: 1371: 1357: 370: 348: 334: 326: 27: 152: 256: 18: 7: 1325: 1323: 172: 1343:. You can help Knowledge (XXG) by 14: 1327: 1390:Drugs not assigned an ATC code 246:, developer of DM4 based drugs 1: 1426: 1322: 1410:Monoclonal antibody stubs 1283: 865:Mirvetuximab soravtansine 265:World Health Organization 183: 26: 1405:Antibody-drug conjugates 304:. In Phillips GL (ed.). 217:(huC242) is linked to a 206:(huC242-SPDB-DM4) is an 1261:Depatuxizumab mafodotin 1202:Tucotuzumab celmoleukin 1153:Rovalpituzumab tesirine 1068:Lorvotuzumab mertansine 958:Clivatuzumab tetraxetan 208:antibody-drug conjugate 1339:–related article is a 1222:Vorsetuzumab mafodotin 1178:Tacatuzumab tetraxetan 983:Denintuzumab mafodotin 928:Bivatuzumab mertansine 855:Loncastuximab tesirine 845:Indatuximab ravtansine 722:Naptumomab estafenatox 1400:Monoclonal antibodies 1207:Vandortuzumab vedotin 1158:Sacituzumab govitecan 1048:Inotuzumab ozogamicin 1033:Gemtuzumab ozogamicin 963:Cofetuzumab pelidotin 943:Cantuzumab ravtansine 938:Cantuzumab mertansine 757:Nofetumomab merpentan 717:Moxetumomab pasudotox 471:Glembatumumab vedotin 357:Monoclonal antibodies 239:Cantuzumab mertansine 227:cantuzumab mertansine 204:Cantuzumab ravtansine 21:Cantuzumab ravtansine 1254:Chimeric + humanized 1058:Lifastuzumab vedotin 918:Belantamab mafodotin 687:Ibritumomab tiuxetan 652:Anatumomab mafenatox 276:WHO Drug Information 1337:monoclonal antibody 1173:Sofituzumab vedotin 1143:Polatuzumab vedotin 1138:Pinatuzumab vedotin 1123:Oportuzumab monatox 953:Citatuzumab bogatox 815:Derlotuximab biotin 800:Brentuximab vedotin 752:Taplitumomab paptox 742:Satumomab pendetide 712:Nacolomab tafenatox 647:Altumomab pentetate 282:(2). Archived from 212:monoclonal antibody 37:Monoclonal antibody 23: 1310:Never to phase III 672:Capromab pendetide 446:Enfortumab vedotin 1352: 1351: 1320: 1319: 1279: 1278: 601:Tisotumab vedotin 315:978-1-4614-5456-4 289:on April 1, 2012. 201: 200: 16:Chemical compound 1417: 1373: 1366: 1359: 1331: 1324: 1232:Rat/mouse hybrid 371: 350: 343: 336: 327: 320: 319: 297: 291: 290: 288: 273: 261: 197: 196: 189: 176: 156: 120: 31: 24: 22: 1425: 1424: 1420: 1419: 1418: 1416: 1415: 1414: 1380: 1379: 1378: 1377: 1321: 1316: 1315: 1300:Clinical trials 1275: 1249: 1226: 889: 776: 630: 360: 354: 324: 323: 316: 299: 298: 294: 286: 271: 263: 262: 258: 253: 235: 219:cytotoxic agent 192: 190: 187:(what is this?) 184: 179: 159: 139: 123: 98: 17: 12: 11: 5: 1423: 1421: 1413: 1412: 1407: 1402: 1397: 1392: 1382: 1381: 1376: 1375: 1368: 1361: 1353: 1350: 1349: 1332: 1318: 1317: 1314: 1313: 1312: 1311: 1308: 1297: 1291: 1285: 1284: 1281: 1280: 1277: 1276: 1274: 1273: 1268: 1266:Duvortuxizumab 1263: 1257: 1255: 1251: 1250: 1248: 1247: 1242: 1236: 1234: 1228: 1227: 1225: 1224: 1219: 1214: 1209: 1204: 1199: 1185: 1180: 1175: 1170: 1165: 1160: 1155: 1150: 1145: 1140: 1135: 1130: 1125: 1120: 1115: 1110: 1105: 1100: 1095: 1090: 1085: 1080: 1075: 1070: 1065: 1060: 1055: 1050: 1045: 1040: 1035: 1030: 1025: 1020: 1015: 1010: 1005: 1000: 995: 990: 985: 980: 975: 970: 965: 960: 955: 950: 945: 940: 935: 933:Brontictuzumab 930: 925: 920: 915: 910: 905: 899: 897: 891: 890: 888: 887: 882: 877: 872: 867: 862: 857: 852: 847: 842: 837: 832: 827: 822: 817: 812: 807: 802: 797: 792: 786: 784: 778: 777: 775: 774: 769: 764: 759: 754: 749: 744: 739: 734: 729: 724: 719: 714: 709: 704: 699: 694: 689: 684: 679: 674: 669: 664: 659: 654: 649: 644: 638: 636: 632: 631: 629: 628: 623: 618: 613: 608: 603: 598: 593: 588: 583: 578: 573: 568: 563: 558: 553: 548: 543: 538: 533: 528: 523: 518: 513: 508: 503: 498: 493: 488: 483: 478: 473: 468: 463: 458: 453: 448: 443: 438: 433: 428: 423: 418: 413: 408: 403: 400:+hyaluronidase 393: 388: 383: 377: 375: 368: 362: 361: 355: 353: 352: 345: 338: 330: 322: 321: 314: 292: 255: 254: 252: 249: 248: 247: 241: 234: 231: 199: 198: 181: 180: 178: 177: 169: 167: 161: 160: 158: 157: 149: 147: 141: 140: 138: 137: 133: 131: 125: 124: 122: 121: 113: 111: 105: 104: 100: 99: 97: 96: 92: 90: 84: 83: 79: 78: 73: 67: 66: 56: 50: 49: 48:Whole antibody 46: 40: 39: 33: 32: 15: 13: 10: 9: 6: 4: 3: 2: 1422: 1411: 1408: 1406: 1403: 1401: 1398: 1396: 1393: 1391: 1388: 1387: 1385: 1374: 1369: 1367: 1362: 1360: 1355: 1354: 1348: 1346: 1342: 1338: 1333: 1330: 1326: 1309: 1307: 1304: 1303: 1301: 1298: 1295: 1292: 1290: 1287: 1286: 1282: 1272: 1269: 1267: 1264: 1262: 1259: 1258: 1256: 1252: 1246: 1243: 1241: 1238: 1237: 1235: 1233: 1229: 1223: 1220: 1218: 1215: 1213: 1210: 1208: 1205: 1203: 1200: 1197: 1193: 1189: 1186: 1184: 1181: 1179: 1176: 1174: 1171: 1169: 1166: 1164: 1161: 1159: 1156: 1154: 1151: 1149: 1148:Rosmantuzumab 1146: 1144: 1141: 1139: 1136: 1134: 1131: 1129: 1126: 1124: 1121: 1119: 1116: 1114: 1111: 1109: 1106: 1104: 1101: 1099: 1096: 1094: 1091: 1089: 1086: 1084: 1081: 1079: 1076: 1074: 1071: 1069: 1066: 1064: 1061: 1059: 1056: 1054: 1051: 1049: 1046: 1044: 1041: 1039: 1036: 1034: 1031: 1029: 1026: 1024: 1021: 1019: 1016: 1014: 1011: 1009: 1006: 1004: 1003:Enoblituzumab 1001: 999: 996: 994: 991: 989: 986: 984: 981: 979: 976: 974: 971: 969: 966: 964: 961: 959: 956: 954: 951: 949: 946: 944: 941: 939: 936: 934: 931: 929: 926: 924: 921: 919: 916: 914: 911: 909: 906: 904: 901: 900: 898: 896: 892: 886: 883: 881: 878: 876: 873: 871: 868: 866: 863: 861: 858: 856: 853: 851: 848: 846: 843: 841: 838: 836: 833: 831: 828: 826: 823: 821: 818: 816: 813: 811: 808: 806: 803: 801: 798: 796: 793: 791: 788: 787: 785: 783: 779: 773: 770: 768: 765: 763: 760: 758: 755: 753: 750: 748: 745: 743: 740: 738: 735: 733: 730: 728: 725: 723: 720: 718: 715: 713: 710: 708: 705: 703: 700: 698: 695: 693: 690: 688: 685: 683: 680: 678: 675: 673: 670: 668: 665: 663: 660: 658: 655: 653: 650: 648: 645: 643: 640: 639: 637: 633: 627: 624: 622: 619: 617: 614: 612: 609: 607: 604: 602: 599: 597: 594: 592: 589: 587: 584: 582: 579: 577: 574: 572: 569: 567: 564: 562: 559: 557: 556:Pembrolizumab 554: 552: 549: 547: 544: 542: 539: 537: 534: 532: 529: 527: 524: 522: 519: 517: 514: 512: 509: 507: 504: 502: 499: 497: 494: 492: 489: 487: 484: 482: 479: 477: 474: 472: 469: 467: 464: 462: 459: 457: 454: 452: 449: 447: 444: 442: 439: 437: 434: 432: 429: 427: 424: 422: 419: 417: 414: 412: 409: 407: 404: 401: 397: 394: 392: 391:Ascrinvacumab 389: 387: 384: 382: 379: 378: 376: 372: 369: 367: 363: 358: 351: 346: 344: 339: 337: 332: 331: 328: 317: 311: 307: 303: 296: 293: 285: 281: 277: 270: 266: 260: 257: 250: 245: 244:ImmunoGen Inc 242: 240: 237: 236: 232: 230: 228: 225:linkage than 224: 220: 216: 213: 209: 205: 195: 188: 182: 175: 171: 170: 168: 166: 162: 155: 151: 150: 148: 146: 142: 135: 134: 132: 130: 126: 119: 115: 114: 112: 110: 106: 101: 94: 93: 91: 89: 85: 82:Clinical data 80: 77: 74: 72: 68: 64: 60: 57: 55: 51: 47: 45: 41: 38: 34: 30: 25: 1345:expanding it 1334: 1163:Sibrotuzumab 1128:Parsatuzumab 1113:Otlertuzumab 1108:Odronextamab 1103:Ocaratuzumab 1098:Obinutuzumab 1073:Lumretuzumab 1028:Flotetuzumab 1023:Ficlatuzumab 1018:Farletuzumab 1013:Etaracizumab 998:Emibetuzumab 942: 885:Zolbetuximab 860:Margetuximab 840:Girentuximab 702:Minretumomab 667:Blinatumomab 606:Teprotumumab 586:Seribantumab 411:Botensilimab 396:Atezolizumab 381:Adecatumumab 305: 295: 284:the original 279: 275: 259: 214: 203: 202: 191:   185:   1296:from market 1271:Ontuxizumab 1245:Ertumaxomab 1240:Catumaxomab 1212:Vanucizumab 1192:+deruxtecan 1188:Trastuzumab 1183:Tigatuzumab 1118:Onartuzumab 1093:Nimotuzumab 1083:Milatuzumab 1053:Labetuzumab 1043:Imgatuzumab 1008:Epcoritamab 993:Emactuzumab 978:Dalotuzumab 968:Dacetuzumab 948:Cirmtuzumab 923:Bevacizumab 908:Alemtuzumab 880:Ublituximab 830:Ensituximab 825:Ecromeximab 820:Dinutuximab 805:Carotuximab 795:Bavituximab 772:Tositumomab 767:Tenatumomab 737:Racotumomab 682:Edrecolomab 657:Arcitumomab 626:Zalutumumab 616:Vantictumab 591:Sugemalimab 581:Robatumumab 576:Rilotumumab 571:Ramucirumab 546:Panitumumab 521:Necitumumab 511:Mapatumumab 506:Lucatumumab 501:Lexatumumab 491:Istiratumab 476:Intetumumab 461:Flanvotumab 456:Figitumumab 441:Dusigitumab 436:Duligotumab 426:Daratumumab 421:Conatumumab 416:Cixutumumab 406:Balstilimab 386:Amivantamab 118:868747-45-9 103:Identifiers 1395:Immunology 1384:Categories 1217:Veltuzumab 1196:+emtansine 1168:Simtuzumab 1133:Pertuzumab 1063:Lintuzumab 1038:Glofitamab 988:Elotuzumab 973:Demcizumab 913:Axatilimab 903:Abituzumab 875:Siltuximab 850:Isatuximab 790:Amatuximab 762:Pintumomab 732:Pemtumomab 727:Oregovomab 662:Bectumomab 642:Abagovomab 596:Tarextumab 566:Radretumab 561:Pritumumab 551:Patritumab 541:Olaratumab 536:Ofatumumab 526:Nesvacumab 516:Narnatumab 486:Iratumumab 481:Ipilimumab 451:Enoticumab 431:Drozitumab 359:for tumors 251:References 215:cantuzumab 154:RNQ8JQ4R9P 129:ChemSpider 109:CAS Number 1306:Phase III 1294:Withdrawn 1088:Naxitamab 1078:Matuzumab 895:Humanized 870:Rituximab 835:Futuximab 810:Cetuximab 747:Solitomab 707:Mitumomab 697:Lilotomab 677:Detumomab 621:Votumumab 611:Tovetumab 531:Nivolumab 496:Icrucumab 466:Ganitumab 223:disulfide 59:Humanized 782:Chimeric 692:Igovomab 267:(2011). 233:See also 194:(verify) 88:ATC code 1289:WHO-EM 312:  174:D10454 71:Target 61:(from 54:Source 1335:This 635:Mouse 374:Human 366:Tumor 287:(PDF) 272:(PDF) 63:mouse 1341:stub 310:ISBN 165:KEGG 145:UNII 136:none 95:none 76:MUC1 44:Type 1386:: 1302:: 1194:/ 280:25 278:. 274:. 229:. 1372:e 1365:t 1358:v 1347:. 1198:) 1190:( 402:) 398:( 349:e 342:t 335:v 318:. 65:)

Index


Monoclonal antibody
Type
Source
Humanized
mouse
Target
MUC1
ATC code
CAS Number
868747-45-9
ChemSpider
UNII
RNQ8JQ4R9P
KEGG
D10454
(what is this?)
(verify)
antibody-drug conjugate
monoclonal antibody
cytotoxic agent
disulfide
cantuzumab mertansine
Cantuzumab mertansine
ImmunoGen Inc
World Health Organization
"International Nonproprietary Names for Pharmaceutical Substances (INN). Proposed INN: List 105"
the original
"Linker technology and impact of linker design on ADC properties."
ISBN

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