1642:
1622:
1610:
1007:
419:
per patient, per year. Gilead maintains that its pricing is comparable to other HIV medications on the market. Elvitegravir/cobicistat/emtricitabine/tenofovir (Stribild) is priced at 39 percent higher than
216:
1191:
1196:
1142:
614:
1581:
171:
778:
382:(a marker of kidney function) may increase with use of elvitegravir/cobicistat/emtricitabine/tenofovir. This is caused by cobicistat's inhibition of tubular secretion in the
1686:
1710:
1148:
1206:
1126:
1211:
1159:
560:
113:
1181:
1165:
1176:
1186:
1453:
1097:
1679:
1552:
1443:
123:
1201:
421:
1725:
1216:
367:
increases the effectiveness of the combination by inhibiting the liver and gut wall enzymes that metabolize elvitegravir. It is taken
772:
553:
429:
1672:
1226:
1110:
490:
424:(Complera), a three-drug HIV regimen approved a year earlier. At the time of Complera's approval, there were concerns about the
1236:
1221:
1001:
981:
899:
884:
872:
201:
81:
1116:
1600:
538:
546:
400:
1569:
1705:
344:
37:
1715:
1393:
1303:
1171:
1132:
436:. HIV drug prices have increased substantially. Atripla, a combination therapy released in 2006, was priced at
1557:
1153:
157:
1231:
491:"Stribild- elvitegravir, cobicistat, emtricitabine, and tenofovir disoproxil fumarate tablet, film coated"
404:
341:
462:"FDA-sourced list of all drugs with black box warnings (Use Download Full Results and View Query links.)"
1720:
1428:
1241:
1121:
991:
590:
28:
1137:
986:
744:
461:
433:
360:
88:
1652:
1246:
1105:
977:
895:
694:
573:
368:
269:
164:
54:
131:
19:
This article is about the combination medication elvitegravir/cobicistat/emtricitabine/tenofovir
1534:
1529:
1388:
1051:
229:
103:
1656:
516:
278:
1413:
69:
1614:
1489:
1448:
608:
440:
per person, per year. Atripla's wholesale prices have risen to the level of
Complera's at
372:
66:
1626:
1563:
1339:
1321:
1284:
569:
1699:
1649:
1329:
1079:
914:
800:
356:
242:
76:
1383:
1373:
954:
944:
762:
719:
714:
709:
671:
651:
581:
352:
184:
179:
49:
1641:
23:. For the combination medication elvitegravir/cobicistat/emtricitabine/tenofovir
1509:
1484:
1423:
1408:
1403:
1067:
1034:
949:
929:
724:
704:
683:
630:
598:
1514:
1494:
1479:
1474:
1438:
1433:
1347:
1292:
1262:
1074:
1062:
1057:
1029:
969:
959:
934:
919:
909:
858:
853:
841:
825:
815:
795:
757:
667:
655:
647:
379:
364:
289:
61:
1524:
1504:
1499:
1469:
1398:
1378:
1311:
1267:
1024:
939:
924:
847:
820:
810:
805:
752:
729:
642:
399:
Elvitegravir/cobicistat/emtricitabine/tenofovir gained approval by the U.S.
117:
1519:
904:
348:
1587:
1418:
964:
734:
383:
1621:
1368:
1363:
314:
678:
637:
625:
305:
251:
223:
542:
236:
662:
577:
469:
1192:
Elvitegravir/cobicistat/emtricitabine/tenofovir alafenamide
210:
142:
1197:
Elvitegravir/cobicistat/emtricitabine/tenofovir disoproxil
407:
for the first time as part of the fixed dose combination.
1143:
Darunavir/cobicistat/emtricitabine/tenofovir alafenamide
1660:
1598:
1462:
1356:
1338:
1320:
1302:
1283:
1276:
1255:
1096:
1043:
1017:
1000:
883:
871:
834:
788:
771:
743:
693:
607:
589:
304:
288:
268:
263:
200:
195:
170:
156:
130:
112:
102:
97:
87:
75:
60:
48:
43:
403:(FDA) in August 2012, for use in adults starting
1149:Dolutegravir/emtricitabine/tenofovir alafenamide
1207:Emtricitabine/rilpivirine/tenofovir alafenamide
1127:Bictegravir/emtricitabine/tenofovir alafenamide
415:Gilead's stated wholesale price of Stribild is
327:Elvitegravir/cobicistat/emtricitabine/tenofovir
277:
38:Elvitegravir/cobicistat/emtricitabine/tenofovir
1212:Emtricitabine/rilpivirine/tenofovir disoproxil
698:(Integrase strand transfer inhibitors (INSTI))
1680:
1160:Dolutegravir/lamivudine/tenofovir alafenamide
554:
8:
1182:Efavirenz/emtricitabine/tenofovir disoproxil
1166:Dolutegravir/lamivudine/tenofovir disoproxil
36:
432:(Atripla), which is marketed by Gilead and
1687:
1673:
1280:
1177:Doravirine/lamivudine/tenofovir disoproxil
1014:
880:
785:
561:
547:
539:
1187:Efavirenz/lamivudine/tenofovir disoproxil
29:Tenofovir alafenamide § combinations
1454:Zinc finger protein transcription factor
1711:Fixed dose combination (antiretroviral)
1605:
453:
363:directly suppress viral reproduction.
35:
122:
7:
1638:
1636:
183:
1202:Emtricitabine/tenofovir alafenamide
422:emtricitabine/rilpivirine/tenofovir
313:
1659:. You can help Knowledge (XXG) by
1217:Emtricitabine/tenofovir disoproxil
14:
430:efavirenz/emtricitabine/tenofovir
1640:
1620:
1608:
1590:. Formerly or rarely used agent.
1227:Lamivudine/nevirapine/zidovudine
1111:Abacavir/dolutegravir/lamivudine
1394:Epigallocatechin gallate (EGCG)
1237:Lamivudine/tenofovir disoproxil
1222:Lamivudine/nevirapine/stavudine
93:Reverse-transcriptase inhibitor
82:Reverse-transcriptase inhibitor
1117:Abacavir/lamivudine/zidovudine
1:
401:Food and Drug Administration
329:, sold under the brand name
992:Tenofovir alafenamide (TAF)
1742:
1635:
987:Tenofovir disoproxil (TDF)
18:
1726:Antiinfective agent stubs
1547:
1008:Discovery and development
779:Discovery and development
615:Discovery and development
521:European Medicines Agency
345:antiretroviral medication
1304:Transcription inhibitors
1256:Pharmacokinetic boosters
1172:Dolutegravir/rilpivirine
1133:Cabotegravir/rilpivirine
773:Protease Inhibitors (PI)
405:antiretroviral treatment
371:. It is manufactured by
16:Combination drug for HIV
1588:initial regimen options
1154:Dolutegravir/lamivudine
631:Enfuvirtide (ENF, T-20)
609:Entry/fusion inhibitors
124:Professional Drug Facts
1429:Portmanteau inhibitors
1322:Translation inhibitors
1232:Lamivudine/raltegravir
1002:Non-nucleoside (NNRTI)
960:Islatravir (EFdA, ISL)
342:fixed-dose combination
1444:Synergistic enhancers
1242:Lamivudine/zidovudine
1122:Atazanavir/cobicistat
1098:Combined formulations
935:Zidovudine (AZT, ZDV)
873:Reverse-transcriptase
745:Maturation inhibitors
347:for the treatment of
1285:Uncoating inhibitors
1138:Darunavir/cobicistat
978:Nucleotide analogues
896:Nucleoside analogues
695:Integrase inhibitors
574:antiretroviral drugs
434:Bristol-Myers Squibb
361:tenofovir disoproxil
333:, also known as the
89:Tenofovir disoproxil
1277:Experimental agents
1247:Lopinavir/ritonavir
1106:Abacavir/lamivudine
1080:Elsulfavirine (ESV)
915:Emtricitabine (FTC)
801:Fosamprenavir (FPV)
497:. 16 September 2021
390:Society and culture
232:(Prescription only)
219:(Prescription only)
55:Integrase inhibitor
40:
1574:Never to phase III
720:Elvitegravir (EVG)
715:Dolutegravir (DTG)
710:Cabotegravir (CAB)
428:wholesale cost of
1706:CYP3A4 inhibitors
1668:
1667:
1596:
1595:
1543:
1542:
1389:Diarylpyrimidines
1092:
1091:
1088:
1087:
1068:Rilpivirine (RPV)
1052:diarylpyrimidines
1035:Delavirdine (DLV)
930:Zalcitabine (ddC)
887:nucleotide (NRTI)
867:
866:
725:Raltegravir (RAL)
705:Bictegravir (BIC)
684:Fostemsavir (FTR)
599:Lenacapavir (LEN)
591:Capsid inhibitors
324:
323:
255:
240:
227:
214:
146:
1733:
1689:
1682:
1675:
1644:
1637:
1625:
1624:
1613:
1612:
1611:
1604:
1414:Hydroxycarbamide
1281:
1075:Doravirine (DOR)
1063:Etravirine (ETR)
1058:Dapivirine (DPV)
1030:Nevirapine (NVP)
1015:
920:Lamivudine (3TC)
910:Didanosine (ddI)
881:
854:Tipranavir (TPV)
842:Atazanavir (ATV)
826:Saquinavir (SQV)
816:Nelfinavir (NFV)
796:Amprenavir (APV)
786:
668:Ibalizumab (IBA)
563:
556:
549:
540:
533:
532:
530:
528:
513:
507:
506:
504:
502:
487:
481:
480:
478:
476:
466:nctr-crs.fda.gov
458:
443:
439:
427:
418:
317:
281:
253:
250:
245:
238:
235:
225:
222:
212:
209:
187:
144:
141:
126:
41:
39:
1741:
1740:
1736:
1735:
1734:
1732:
1731:
1730:
1716:Gilead Sciences
1696:
1695:
1694:
1693:
1633:
1631:
1619:
1609:
1607:
1599:
1597:
1592:
1591:
1579:
1564:Clinical trials
1539:
1490:Dexelvucitabine
1458:
1449:Tre recombinase
1352:
1334:
1316:
1312:Tat antagonists
1298:
1272:
1251:
1084:
1039:
1025:Efavirenz (EFV)
1004:
996:
925:Stavudine (d4T)
886:
874:
863:
848:Darunavir (DRV)
830:
821:Ritonavir (RTV)
811:Lopinavir (LPV)
806:Indinavir (IDV)
775:
767:
739:
697:
689:
643:Maraviroc (MVC)
611:
603:
585:
570:Antiviral drugs
567:
537:
536:
526:
524:
517:"Stribild EPAR"
515:
514:
510:
500:
498:
489:
488:
484:
474:
472:
460:
459:
455:
450:
441:
437:
425:
416:
413:
397:
392:
373:Gilead Sciences
320:
300:
284:
259:
243:
191:
159:
152:
133:
67:Cytochrome P450
32:
17:
12:
11:
5:
1739:
1737:
1729:
1728:
1723:
1718:
1713:
1708:
1698:
1697:
1692:
1691:
1684:
1677:
1669:
1666:
1665:
1645:
1630:
1629:
1617:
1594:
1593:
1578:
1577:
1576:
1575:
1572:
1561:
1555:
1549:
1548:
1545:
1544:
1541:
1540:
1538:
1537:
1532:
1527:
1522:
1517:
1512:
1507:
1502:
1497:
1492:
1487:
1482:
1477:
1472:
1466:
1464:
1460:
1459:
1457:
1456:
1451:
1446:
1441:
1436:
1431:
1426:
1421:
1416:
1411:
1406:
1401:
1396:
1391:
1386:
1381:
1376:
1371:
1366:
1360:
1358:
1354:
1353:
1351:
1350:
1344:
1342:
1336:
1335:
1333:
1332:
1326:
1324:
1318:
1317:
1315:
1314:
1308:
1306:
1300:
1299:
1297:
1296:
1289:
1287:
1278:
1274:
1273:
1271:
1270:
1265:
1263:Cobicistat (c)
1259:
1257:
1253:
1252:
1250:
1249:
1244:
1239:
1234:
1229:
1224:
1219:
1214:
1209:
1204:
1199:
1194:
1189:
1184:
1179:
1174:
1169:
1163:
1157:
1151:
1146:
1140:
1135:
1130:
1124:
1119:
1114:
1108:
1102:
1100:
1094:
1093:
1090:
1089:
1086:
1085:
1083:
1082:
1077:
1072:
1071:
1070:
1065:
1060:
1047:
1045:
1041:
1040:
1038:
1037:
1032:
1027:
1021:
1019:
1012:
998:
997:
995:
994:
989:
973:
972:
967:
962:
957:
952:
947:
942:
937:
932:
927:
922:
917:
912:
907:
905:Abacavir (ABC)
891:
889:
885:Nucleoside and
878:
869:
868:
865:
864:
862:
861:
856:
851:
845:
838:
836:
832:
831:
829:
828:
823:
818:
813:
808:
803:
798:
792:
790:
783:
769:
768:
766:
765:
760:
755:
749:
747:
741:
740:
738:
737:
732:
727:
722:
717:
712:
707:
701:
699:
691:
690:
688:
687:
675:
659:
645:
634:
621:
619:
605:
604:
602:
601:
595:
593:
587:
586:
568:
566:
565:
558:
551:
543:
535:
534:
523:. 13 June 2013
508:
482:
452:
451:
449:
446:
412:
409:
396:
393:
391:
388:
322:
321:
319:
318:
310:
308:
302:
301:
299:
298:
294:
292:
286:
285:
283:
282:
274:
272:
266:
265:
261:
260:
258:
257:
248:
233:
220:
206:
204:
198:
197:
193:
192:
190:
189:
176:
174:
168:
167:
162:
160:administration
154:
153:
151:
150:
148:
138:
136:
128:
127:
120:
110:
109:
106:
100:
99:
95:
94:
91:
85:
84:
79:
73:
72:
64:
58:
57:
52:
46:
45:
44:Combination of
15:
13:
10:
9:
6:
4:
3:
2:
1738:
1727:
1724:
1722:
1719:
1717:
1714:
1712:
1709:
1707:
1704:
1703:
1701:
1690:
1685:
1683:
1678:
1676:
1671:
1670:
1664:
1662:
1658:
1655:article is a
1654:
1651:
1650:antiinfective
1646:
1643:
1639:
1634:
1628:
1623:
1618:
1616:
1606:
1602:
1589:
1586:
1583:
1573:
1571:
1568:
1567:
1565:
1562:
1559:
1556:
1554:
1551:
1550:
1546:
1536:
1533:
1531:
1528:
1526:
1523:
1521:
1518:
1516:
1513:
1511:
1508:
1506:
1503:
1501:
1498:
1496:
1493:
1491:
1488:
1486:
1483:
1481:
1478:
1476:
1473:
1471:
1468:
1467:
1465:
1463:Failed agents
1461:
1455:
1452:
1450:
1447:
1445:
1442:
1440:
1437:
1435:
1432:
1430:
1427:
1425:
1422:
1420:
1417:
1415:
1412:
1410:
1407:
1405:
1402:
1400:
1397:
1395:
1392:
1390:
1387:
1385:
1382:
1380:
1377:
1375:
1372:
1370:
1367:
1365:
1362:
1361:
1359:
1355:
1349:
1346:
1345:
1343:
1341:
1337:
1331:
1330:Trichosanthin
1328:
1327:
1325:
1323:
1319:
1313:
1310:
1309:
1307:
1305:
1301:
1294:
1291:
1290:
1288:
1286:
1282:
1279:
1275:
1269:
1268:Ritonavir (r)
1266:
1264:
1261:
1260:
1258:
1254:
1248:
1245:
1243:
1240:
1238:
1235:
1233:
1230:
1228:
1225:
1223:
1220:
1218:
1215:
1213:
1210:
1208:
1205:
1203:
1200:
1198:
1195:
1193:
1190:
1188:
1185:
1183:
1180:
1178:
1175:
1173:
1170:
1167:
1164:
1161:
1158:
1155:
1152:
1150:
1147:
1144:
1141:
1139:
1136:
1134:
1131:
1128:
1125:
1123:
1120:
1118:
1115:
1112:
1109:
1107:
1104:
1103:
1101:
1099:
1095:
1081:
1078:
1076:
1073:
1069:
1066:
1064:
1061:
1059:
1056:
1055:
1054:
1053:
1049:
1048:
1046:
1042:
1036:
1033:
1031:
1028:
1026:
1023:
1022:
1020:
1016:
1013:
1011:
1009:
1003:
999:
993:
990:
988:
985:
983:
979:
975:
974:
971:
968:
966:
963:
961:
958:
956:
953:
951:
948:
946:
943:
941:
938:
936:
933:
931:
928:
926:
923:
921:
918:
916:
913:
911:
908:
906:
903:
901:
897:
893:
892:
890:
888:
882:
879:
876:
870:
860:
857:
855:
852:
849:
846:
843:
840:
839:
837:
833:
827:
824:
822:
819:
817:
814:
812:
809:
807:
804:
802:
799:
797:
794:
793:
791:
787:
784:
782:
780:
774:
770:
764:
761:
759:
756:
754:
751:
750:
748:
746:
742:
736:
733:
731:
728:
726:
723:
721:
718:
716:
713:
711:
708:
706:
703:
702:
700:
696:
692:
685:
681:
680:
676:
673:
669:
665:
664:
660:
657:
653:
649:
646:
644:
640:
639:
635:
632:
628:
627:
623:
622:
620:
618:
616:
610:
606:
600:
597:
596:
594:
592:
588:
583:
579:
576:used against
575:
571:
564:
559:
557:
552:
550:
545:
544:
541:
522:
518:
512:
509:
496:
492:
486:
483:
471:
467:
463:
457:
454:
447:
445:
435:
431:
423:
410:
408:
406:
402:
394:
389:
387:
385:
381:
376:
374:
370:
366:
362:
358:
357:emtricitabine
354:
350:
346:
343:
339:
336:
332:
328:
316:
312:
311:
309:
307:
303:
296:
295:
293:
291:
287:
280:
276:
275:
273:
271:
267:
262:
256: Rx-only
249:
246:
234:
231:
221:
218:
208:
207:
205:
203:
199:
194:
186:
181:
178:
177:
175:
173:
169:
166:
163:
161:
155:
149:
140:
139:
137:
135:
129:
125:
121:
119:
115:
111:
107:
105:
101:
98:Clinical data
96:
92:
90:
86:
83:
80:
78:
77:Emtricitabine
74:
71:
68:
65:
63:
59:
56:
53:
51:
47:
42:
34:
30:
26:
22:
1721:Hepatotoxins
1661:expanding it
1647:
1632:
1584:
1384:Cyanovirin-N
1374:Calanolide A
1050:
1044:2 generation
1018:1 generation
1005:
976:
955:Elvucitabine
945:Apricitabine
894:
835:2 generation
789:1 generation
776:
763:Fipravirimat
677:
672:Semzuvolimab
661:
652:Cenicriviroc
636:
624:
612:
525:. Retrieved
520:
511:
499:. Retrieved
494:
485:
473:. Retrieved
465:
456:
414:
398:
395:Legal status
377:
353:Elvitegravir
337:
334:
330:
326:
325:
279:1430117-57-9
202:Legal status
196:Legal status
50:Elvitegravir
33:
24:
20:
1585:recommended
1560:from market
1510:Lersivirine
1485:Capravirine
1424:Miltefosine
1409:Griffithsin
1404:Fosdevirine
950:Censavudine
580:(primarily
264:Identifiers
104:Trade names
25:alafenamide
1700:Categories
1515:Lodenosine
1495:Droxinavir
1480:Brecanavir
1475:Atevirdine
1439:Seliciclib
1434:Scytovirin
1348:Elipovimab
1293:TRIM5alpha
970:Stampidine
875:inhibitors
859:TMC-310911
758:BMS-955176
656:Leronlimab
648:Vicriviroc
475:22 October
448:References
442:US$ 20,500
438:US$ 13,800
426:US$ 20,500
417:US$ 28,500
380:creatinine
365:Cobicistat
290:ChemSpider
270:CAS Number
62:Cobicistat
21:disoproxil
1570:Phase III
1558:Withdrawn
1535:Telinavir
1530:Palinavir
1525:Mozenavir
1505:Emivirine
1500:Lasinavir
1470:Aplaviroc
1399:Foscarnet
1379:Ceragenin
940:Amdoxovir
753:Bevirimat
730:BI 224436
411:Economics
158:Routes of
132:Pregnancy
118:Drugs.com
70:inhibitor
1615:Medicine
1520:Loviride
495:DailyMed
369:by mouth
349:HIV/AIDS
331:Stribild
172:ATC code
165:By mouth
147: B3
134:category
108:Stribild
1627:Viruses
1601:Portals
1419:KP-1461
965:Racivir
735:MK-2048
527:24 July
501:24 July
384:nephron
340:, is a
247:Rx-only
244:WARNING
188:)
182: (
180:J05AR09
1553:WHO-EM
1369:BIT225
1364:Abzyme
1295:(gene)
982:NtRTIs
877:(RTIs)
378:Serum
315:D10756
241:
228:
215:
27:, see
1648:This
1357:Other
1340:BNAbs
900:NRTIs
679:gp120
1657:stub
1653:drug
1582:DHHS
638:CCR5
626:gp41
529:2024
503:2024
477:2023
359:and
338:pill
335:Quad
306:KEGG
297:none
114:AHFS
663:CD4
582:J05
578:HIV
470:FDA
230:POM
185:WHO
1702::
1566::
670:,
654:,
650:,
572::
519:.
493:.
468:.
464:.
444:.
386:.
375:.
355:,
351:.
252:EU
237:US
224:UK
217:S4
211:AU
143:AU
1688:e
1681:t
1674:v
1663:.
1603::
1580:°
1168:°
1162:°
1156:°
1145:°
1129:°
1113:°
1010:)
1006:(
984::
980:/
902::
898:/
850:°
844:°
781:)
777:(
686:)
682:(
674:)
666:(
658:)
641:(
633:)
629:(
617:)
613:(
584:)
562:e
555:t
548:v
531:.
505:.
479:.
254::
239::
226::
213::
145::
116:/
31:.
Text is available under the Creative Commons Attribution-ShareAlike License. Additional terms may apply.