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for all of the aforementioned indications before being discontinued due to the observation of possible predictive signs of
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InChI=1S/C15H13FN2/c1-10-8-11(2)18-14(15(10)17)7-6-12-4-3-5-13(16)9-12/h3-5,8-9H,17H2,1-2H3
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Benign and
Neoplastic Conditions of the Esophagus, An Issue of Gastroenterology Clinics
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Development of ADX10059 Ended for Long-term Use - Addex
Therapeutics
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501:. Springer Science & Business Media. pp. 120–.
474:. Springer Science & Business Media. pp. 397–.
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Célanire S, Duvey G, Poli S, Rocher JP (January 2012).
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1700:Glutamate receptor negative allosteric modulators
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1591:Glutamate metabolism/transport modulators
1498:Tooltip Metabotropic glutamate receptor 8
1399:Tooltip Metabotropic glutamate receptor 7
1327:Tooltip Metabotropic glutamate receptor 6
1223:Tooltip Metabotropic glutamate receptor 4
1074:Tooltip Metabotropic glutamate receptor 3
916:Tooltip Metabotropic glutamate receptor 2
730:Tooltip Metabotropic glutamate receptor 5
616:Tooltip Metabotropic glutamate receptor 1
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1587:Ionotropic glutamate receptor modulators
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468:Stein MB, Steckler T (30 July 2010).
422:Annual Reports in Medicinal Chemistry
7:
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1130:Pomaglumetad methionil (LY-2140023)
982:Pomaglumetad methionil (LY-2140023)
106:
1628:. You can help Knowledge (XXG) by
14:
1608:
495:Dominguez C (18 November 2010).
373:in patients with long-term use.
224:
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1526:Positive allosteric modulators:
1477:Negative allosteric modulators:
1266:Positive allosteric modulators:
1184:Negative allosteric modulators:
1048:Negative allosteric modulators:
991:Positive allosteric modulators:
847:Negative allosteric modulators:
790:Positive allosteric modulators:
588:Metabotropic glutamate receptor
356:gastroesophageal reflux disease
346:which was under development by
305:Key:MEDCLNYIYBERKO-UHFFFAOYSA-N
1675:Drugs not assigned an ATC code
209:
73:2--4,6-dimethyl-3-pyridinamine
1:
1583:Receptor/signaling modulators
328:negative allosteric modulator
280:Fc2cccc(C#Cc1nc(cc(c1N)C)C)c2
522:Shaheen NJ (25 March 2013).
1721:
1680:MGlu5 receptor antagonists
1603:
498:Neurodegenerative Diseases
199:Chemical and physical data
1705:Nervous system drug stubs
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1115:LY-404,039 (pomaglumetad)
962:LY-404,039 (pomaglumetad)
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1620:article relating to the
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350:for the treatment of
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34:
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1630:expanding it
1615:
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1536:Antagonists:
1535:
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1505:
1476:
1435:Antagonists:
1434:
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1353:Antagonists:
1352:
1334:
1281:Antagonists:
1280:
1265:
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1142:Antagonists:
1141:
1135:Talaglumetad
1081:
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1001:Antagonists:
1000:
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987:Talaglumetad
923:
884:
860:Dipraglurant
855:Basimglurant
846:
800:Antagonists:
799:
789:
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679:Antagonists:
678:
623:
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517:
497:
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470:
449:. Retrieved
440:
421:
411:
388:Dipraglurant
383:Basimglurant
323:
315:
314:
1262:VU-0155,041
1187:Decoglurant
1051:Decoglurant
885:Raseglurant
833:Remeglurant
818:Mavoglurant
682:BAY 36-7620
398:Mavoglurant
316:Raseglurant
242: g·mol
92:757950-09-7
57:Identifiers
21:Raseglurant
1669:Categories
1529:AZ12216052
1269:Foliglurax
1257:VU-001,171
1170:LY-341,495
1165:LY-307,452
1120:LY-487,379
1110:LY-379,268
1029:LY-341,495
1024:LY-307,452
972:LY-566,332
967:LY-487,379
957:LY-379,268
813:LY-344,545
793:LSN2463359
702:LY-456,236
697:LY-367,385
591:modulators
451:2017-04-05
404:References
340:derivative
247:3D model (
235:Molar mass
157:66UCJ8Z8L1
128:ChemSpider
83:CAS Number
66:IUPAC name
1580:See also:
1514:Glutamate
1506:Agonists:
1428:LSP2-9166
1415:Glutamate
1407:Agonists:
1338:Glutamate
1335:Agonists:
1247:LSP2-9166
1234:Glutamate
1231:Agonists:
1206:Group III
1192:RO4491533
1100:Glutamate
1095:Eglumegad
1082:Agonists:
1056:RO4491533
947:Glutamate
942:Eglumegad
924:Agonists:
771:Glutamate
746:ADX-47273
738:Agonists:
662:Ro67-7476
657:Ro67-4853
652:Ro01-6128
637:Glutamate
624:Agonists:
324:ADX-10059
1564:UBP-1112
1480:ADX71743
1468:UBP-1112
1381:UBP-1112
1309:UBP-1112
1180:MGS-0039
1125:MGS-0028
1039:MGS-0039
977:MGS-0028
899:Group II
843:SIB-1893
838:SIB-1757
828:NPS-2390
712:NPS-2390
672:Theanine
377:See also
364:phase II
352:migraine
336:receptor
117:10331863
42:ATC code
870:GRN-529
865:Fenobam
850:AZD9272
786:VU-1545
687:CPCCOEt
599:Group I
393:Fenobam
330:of the
326:) is a
240:240.281
205:Formula
137:8507323
103:PubChem
1473:XAP044
1410:AMN082
1090:DCG-IV
1085:CBiPES
1044:PCCG-4
937:DCG-IV
932:CBiPES
532:
505:
478:
428:
358:, and
273:SMILES
1624:is a
1616:This
1491:mGluR
1448:MMPIP
1392:mGluR
1320:mGluR
1252:PHCCC
1216:mGluR
1160:HYDIA
1150:CECXG
1145:APICA
1067:mGluR
1019:HYDIA
1009:CECXG
1004:APICA
909:mGluR
808:DMeOB
751:CDPPB
723:mGluR
667:VU-71
609:mGluR
293:InChI
249:JSmol
1626:stub
1618:drug
1559:MTPG
1554:MSOP
1549:MPPG
1544:MAP4
1539:CPPG
1522:-AP4
1509:DCPG
1463:MTPG
1458:MSOP
1453:MPPG
1443:MAP4
1438:CPPG
1423:-AP4
1376:MTPG
1371:MSOP
1366:MPPG
1361:MAP4
1356:CPPG
1346:-AP4
1304:MTPG
1299:MSOP
1294:MPPG
1289:MAP4
1284:CPPG
1274:MPEP
1242:-AP4
1175:MCPG
1155:EGLU
1034:MCPG
1014:EGLU
927:BINA
880:MTEP
875:MPEP
823:MCPG
803:CTEP
766:DHPG
756:CHPG
741:ACPD
707:MCPG
632:DHPG
627:ACPD
530:ISBN
503:ISBN
476:ISBN
426:ISBN
344:MPEP
338:and
332:mGlu
148:UNII
49:None
761:DFB
342:of
320:INN
173:EPA
107:CID
1671::
1589:•
1585:•
1524:;
1475:;
1264:;
1182:;
1046:;
989:;
845:;
788:;
460:^
420:.
354:,
219:13
213:15
1657:e
1650:t
1643:v
1632:.
1520:L
1493:8
1421:L
1394:7
1344:L
1322:6
1240:L
1218:4
1069:3
911:2
725:5
611:1
580:e
573:t
566:v
538:.
511:.
484:.
454:.
434:.
334:5
318:(
251:)
228:2
225:N
222:F
216:H
210:C
175:)
171:(
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