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Template:Composition of conjugated estrogens and properties of constituents

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Bhavnani BR, Tam SP, Lu X (October 2008). "Structure activity relationships and differential interactions and functional activity of various equine estrogens mediated via estrogen receptors (ERs) ERalpha and ERbeta".
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Bhavnani BR, Stanczyk FZ (July 2014). "Pharmacology of conjugated equine estrogens: efficacy, safety and mechanism of action".
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All listed compounds are present in conjugated estrogen products specifically in the form of the
256: 645: 607: 580: 543: 537: 515: 497:"Pharmacology of estrogens and progestogens: influence of different routes of administration" 637: 572: 507: 459: 228: 663: 576: 511: 284: 649: 584: 519: 641: 463: 172: 456: 75: 66: 102: 91: 466: 469:(i.e., as sodium estrone sulfate, sodium equilin sulfate, etc.). 606:(36th ed.). London: Pharmaceutical Press. p. 2087. 542:. Lippincott Williams & Wilkins. pp. 751–. 539:Clinical Gynecologic Endocrinology and Infertility 531: 529: 110: 97: 82: 490: 488: 536:Marc A. Fritz; Leon Speroff (28 March 2012). 28: 8: 35: 21: 15: 675:Templates that generate named references 604:Martindale: The Complete Drug Reference 484: 450: 16: 7: 600:"Sex hormones and their modulators" 14: 87:Tooltip Relative binding affinity 598:Sweetman, Sean C., ed. (2009). 46:and properties of constituents 1: 565:J. Steroid Biochem. Mol. Biol 577:10.1016/j.jsbmb.2013.10.011 691: 512:10.1080/13697130500148875 451: 670:Medication templates 642:10.1210/en.2008-0304 397:17β-Dihydroequilenin 341:17α-Dihydroequilenin 118:Conjugated estrogens 44:conjugated estrogens 506:. 8 Suppl 1: 3–63. 47: 313:17β-Dihydroequilin 201:17α-Dihydroequilin 613:978-0-85369-840-1 549:978-1-4511-4847-3 476: 475: 682: 654: 653: 624: 618: 617: 595: 589: 588: 560: 554: 553: 533: 524: 523: 501: 492: 112: 99: 88: 84: 72:Relative potency 48: 37: 30: 23: 690: 689: 685: 684: 683: 681: 680: 679: 660: 659: 658: 657: 636:(10): 4857–70. 626: 625: 621: 614: 597: 596: 592: 562: 561: 557: 550: 535: 534: 527: 499: 495:Kuhl H (2005). 494: 493: 486: 481: 425:Δ-17β-Estradiol 401:Δ-17β-Estradiol 345:Δ-17α-Estradiol 317:Δ-17β-Estradiol 205:Δ-17α-Estradiol 109: 101: 90: 86: 73: 64: 42:Composition of 41: 12: 11: 5: 688: 686: 678: 677: 672: 662: 661: 656: 655: 619: 612: 590: 555: 548: 525: 483: 482: 480: 477: 474: 473: 449: 448: 445: 442: 439: 436: 433: 430: 427: 421: 420: 417: 414: 411: 408: 405: 402: 399: 393: 392: 389: 386: 383: 380: 377: 374: 371: 365: 364: 361: 358: 355: 352: 349: 346: 343: 337: 336: 333: 330: 327: 324: 321: 318: 315: 309: 308: 305: 302: 299: 296: 293: 290: 287: 281: 280: 277: 274: 271: 268: 265: 262: 259: 253: 252: 249: 246: 243: 240: 237: 234: 231: 225: 224: 221: 218: 215: 212: 209: 206: 203: 197: 196: 193: 190: 187: 184: 181: 178: 175: 169: 168: 165: 162: 159: 156: 153: 150: 147: 141: 140: 137: 134: 131: 128: 125: 122: 119: 115: 114: 106: 95: 79: 70: 58: 57:Proportion (%) 55: 52: 40: 39: 32: 25: 17: 13: 10: 9: 6: 4: 3: 2: 687: 676: 673: 671: 668: 667: 665: 651: 647: 643: 639: 635: 631: 630:Endocrinology 623: 620: 615: 609: 605: 601: 594: 591: 586: 582: 578: 574: 570: 566: 559: 556: 551: 545: 541: 540: 532: 530: 526: 521: 517: 513: 509: 505: 498: 491: 489: 485: 478: 472: 468: 465: 461: 458: 454: 446: 443: 440: 437: 434: 432:Small amounts 431: 428: 426: 423: 422: 418: 415: 412: 409: 406: 403: 400: 398: 395: 394: 390: 387: 384: 381: 378: 375: 372: 370: 369:17β-Estradiol 367: 366: 362: 359: 356: 353: 350: 347: 344: 342: 339: 338: 334: 331: 328: 325: 322: 319: 316: 314: 311: 310: 306: 303: 300: 297: 294: 291: 288: 286: 283: 282: 278: 275: 272: 269: 266: 263: 260: 258: 255: 254: 250: 247: 244: 241: 238: 235: 232: 230: 229:17α-Estradiol 227: 226: 222: 219: 216: 213: 210: 207: 204: 202: 199: 198: 194: 191: 188: 185: 182: 179: 176: 174: 171: 170: 166: 163: 160: 157: 154: 151: 148: 146: 143: 142: 138: 135: 132: 129: 126: 123: 120: 117: 116: 107: 104: 96: 93: 85: 80: 77: 71: 68: 63: 59: 56: 53: 50: 49: 45: 38: 33: 31: 26: 24: 19: 18: 633: 629: 622: 603: 593: 568: 564: 558: 538: 503: 470: 452: 20: 504:Climacteric 664:Categories 479:References 307:0.50–0.75 571:: 16–29. 289:Δ-Estrone 285:Equilenin 257:Δ-Estrone 208:13.5–19.5 180:22.4–30.5 177:Δ-Estrone 152:49.1–61.5 108:ERα / ERβ 60:Relative 650:18599548 585:24176763 520:16112947 471:Sources: 376:0.56–0.9 51:Compound 464:sulfate 462:of the 404:0.5–0.7 348:1.2–1.6 320:0.5–4.0 292:2.2–2.8 264:3.5–3.9 236:2.5–9.5 173:Equilin 145:Estrone 74:in the 65:in the 62:potency 54:Synonym 648:  610:  583:  546:  518:  467:esters 457:sodium 453:Notes: 113:ratio 76:uterus 67:vagina 500:(PDF) 460:salts 447:0.94 419:0.75 391:1.00 363:0.40 351:0.018 335:1.05 304:20–29 279:0.60 251:0.45 223:1.30 195:0.26 167:0.50 646:PMID 608:ISBN 581:PMID 544:ISBN 516:PMID 407:0.21 298:11.4 239:0.11 211:0.06 638:doi 634:149 573:doi 569:142 508:doi 410:9.4 388:100 385:100 379:100 354:1.3 332:108 329:113 326:200 295:1.3 242:3.5 214:2.6 130:100 124:100 111:RBA 105:(%) 103:ERβ 100:for 98:RBA 94:(%) 92:ERα 89:for 83:RBA 78:(%) 69:(%) 666:: 644:. 632:. 602:. 579:. 567:. 528:^ 514:. 502:. 487:^ 444:72 441:68 416:90 413:68 360:49 357:20 323:83 301:15 276:32 273:19 248:42 245:19 220:32 217:41 192:49 189:13 186:80 183:42 164:52 161:26 158:32 155:30 139:– 127:38 652:. 640:: 616:. 587:. 575:: 552:. 522:. 510:: 438:? 435:? 429:– 382:? 373:– 270:? 267:? 261:– 233:– 149:– 136:– 133:– 121:– 36:e 29:t 22:v

Index

v
t
e
conjugated estrogens
potency
vagina
uterus
RBA
ERα
ERβ
Estrone
Equilin
17α-Dihydroequilin
17α-Estradiol
Δ-Estrone
Equilenin
17β-Dihydroequilin
17α-Dihydroequilenin
17β-Estradiol
17β-Dihydroequilenin
Δ-17β-Estradiol
sodium
salts
sulfate
esters


"Pharmacology of estrogens and progestogens: influence of different routes of administration"
doi
10.1080/13697130500148875

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