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243:. The interaction with the nociceptin receptor is expected to block the abuse and dependence-related side effects that are typical of opioids. A study in nonhuman primates found that AT-121 has morphine-like analgesic effects, but suppressed the addictive effects.
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Ding H, Kiguchi N, Yasuda D, Daga PR, Polgar WE, Lu JJ, et al. (August 2018).
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CC(C)1CC(CC1)N1CCC2(CC1)C(=O)N(CCNS(N)(=O)=O)CC1=CC=CC=C21
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231:. It was designed to be bifunctional, acting as an
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387:. You can help Knowledge (XXG) by
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342:. Science Daily. August 29, 2018.
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42:Legal status
36:Legal status
263:Oliceridine
176: g·mol
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381:analgesic
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