Knowledge (XXG)

Quilizumab

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1613: 410:
Gauvreau GM, Harris JM, Boulet LP, Scheerens H, Fitzgerald JM, Putnam WS, Cockcroft DW, Davis BE, Leigh R, Zheng Y, Dahlén B, Wang Y, Maciuca R, Mayers I, Liao XC, Wu LC, Matthews JG, O'Byrne PM (July 2014). "Targeting membrane-expressed IgE B cell receptor with an antibody to the M1 prime epitope
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Harris JM, Cabanski CR, Scheerens H, Samineni D, Bradley MS, Cochran C, Staubach P, Metz M, Sussman G, Maurer M (December 2016). "A randomized trial of quilizumab in adults with refractory chronic spontaneous urticaria".
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Harris JM, Maciuca R, Bradley MS, Cabanski CR, Scheerens H, Lim J, Cai F, Kishnani M, Liao XC, Samineni D, Zhu R, Cochran C, Soong W, Diaz JD, Perin P, Tsukayama M, Dimov D, Agache I, Kelsen SG (March 2016).
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Deza G, Ricketti PA, Giménez-Arnau AM, Casale TB (2018). "Emerging Biomarkers and Therapeutic Pipelines for Chronic Spontaneous Urticaria".
1693: 1640: 241: 1678: 1544: 1554: 279: 135: 1589: 297: 361:"A randomized trial of the efficacy and safety of quilizumab in adults with inadequately controlled allergic asthma" 1138: 293: 1577: 650: 572: 854: 1620: 99: 44: 27: 1039: 998: 838: 630: 528: 436: 298:"International Nonproprietary Names for Pharmaceutical Substances (INN). Proposed INN: List 106" 930: 600: 541: 520: 485: 428: 392: 340: 1624: 108: 920: 910: 512: 475: 467: 420: 382: 372: 332: 274: 180: 144: 1338: 1114: 454:
Licari A, Castagnoli R, Panfili E, Marseglia A, Brambilla I, Marseglia GL (March 2017).
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Statement On A Nonproprietary Name Adopted By The USAN Council - Quilizumab
20: 822: 745: 655: 625: 1299: 1184: 61: 1524: 245: 244:) is a humanized monoclonal antibody designed for the treatment of 164: 53: 456:"An Update on Anti-IgE Therapy in Pediatric Respiratory Diseases" 249: 155: 66: 545: 1628: 1532: 1522: 1502: 1431: 1365: 1356: 1325: 997: 929: 863: 592: 583: 218: 179: 174: 154: 134: 118: 98: 93: 77: 72: 60: 43: 33: 26: 107: 1648: 557: 8: 19: 1655: 1641: 1529: 1362: 589: 564: 550: 542: 479: 386: 376: 143: 267: 18: 7: 1684:Drugs developed by Hoffmann-La Roche 1609: 1607: 163: 1627:. You can help Knowledge (XXG) by 14: 472:10.2174/1573398X13666170616110738 1611: 197: 191: 1674:Drugs not assigned an ATC code 209: 203: 185: 1: 1689:Drugs developed by Genentech 505:J Allergy Clin Immunol Pract 425:10.1126/scitranslmed.3008961 280:American Medical Association 255:This drug was developed by 1710: 1606: 517:10.1016/j.jaip.2018.02.024 337:10.1016/j.jaci.2016.06.023 175:Chemical and physical data 1694:Monoclonal antibody stubs 1567: 411:reduces IgE production". 378:10.1186/s12931-016-0347-2 294:World Health Organization 325:J. Allergy Clin. Immunol 1623:–related article is a 1679:Monoclonal antibodies 651:Camidanlumab tesirine 573:Monoclonal antibodies 1326:Chimeric + humanized 855:Nivolumab/relatlimab 305:WHO Drug Information 1621:monoclonal antibody 460:Curr Respir Med Rev 28:Monoclonal antibody 23: 16:Monoclonal antibody 1594:Never to phase III 1040:Certolizumab pegol 1007:Immunosuppressive: 1636: 1635: 1604: 1603: 1563: 1562: 1518: 1517: 1352: 1351: 1307:Immune activation 799:Immune activation 601:Immunosuppression 235: 234: 1701: 1657: 1650: 1643: 1615: 1608: 1530: 1363: 921:Zolimomab aritox 911:Telimomab aritox 590: 566: 559: 552: 543: 537: 536: 511:(4): 1108–1117. 500: 494: 493: 483: 451: 445: 444: 419:(243): 243ra85. 407: 401: 400: 390: 380: 355: 349: 348: 331:(6): 1730–1732. 319: 313: 312: 302: 290: 284: 272: 230: 228: 211: 205: 199: 193: 187: 167: 147: 111: 24: 22: 1709: 1708: 1704: 1703: 1702: 1700: 1699: 1698: 1664: 1663: 1662: 1661: 1605: 1600: 1599: 1584:Clinical trials 1559: 1514: 1498: 1427: 1348: 1339:Rozanolixizumab 1327: 1321: 1313: 1302: 1115:Lulizumab pegol 993: 925: 859: 579: 570: 540: 502: 501: 497: 453: 452: 448: 409: 408: 404: 357: 356: 352: 321: 320: 316: 300: 292: 291: 287: 273: 269: 265: 226: 224: 214: 208: 202: 196: 190: 170: 150: 130: 114: 89: 17: 12: 11: 5: 1707: 1705: 1697: 1696: 1691: 1686: 1681: 1676: 1666: 1665: 1660: 1659: 1652: 1645: 1637: 1634: 1633: 1616: 1602: 1601: 1598: 1597: 1596: 1595: 1592: 1581: 1575: 1569: 1568: 1565: 1564: 1561: 1560: 1558: 1557: 1552: 1547: 1542: 1536: 1534: 1527: 1520: 1519: 1516: 1515: 1513: 1512: 1506: 1504: 1500: 1499: 1497: 1496: 1491: 1486: 1481: 1476: 1471: 1466: 1461: 1456: 1451: 1446: 1441: 1435: 1433: 1429: 1428: 1426: 1425: 1420: 1415: 1410: 1405: 1400: 1395: 1390: 1385: 1380: 1375: 1369: 1367: 1360: 1354: 1353: 1350: 1349: 1347: 1346: 1341: 1336: 1330: 1328: 1323: 1322: 1304: 1303: 1297: 1292: 1287: 1282: 1277: 1272: 1267: 1262: 1257: 1252: 1247: 1242: 1237: 1232: 1227: 1222: 1217: 1212: 1207: 1202: 1197: 1192: 1187: 1182: 1177: 1172: 1167: 1162: 1157: 1152: 1147: 1142: 1139:+hyaluronidase 1132: 1127: 1122: 1117: 1112: 1107: 1102: 1097: 1092: 1087: 1082: 1077: 1072: 1067: 1062: 1057: 1052: 1047: 1042: 1037: 1032: 1027: 1022: 1017: 1012: 1003: 1001: 995: 994: 992: 991: 986: 981: 976: 971: 966: 961: 956: 951: 946: 941: 935: 933: 927: 926: 924: 923: 918: 913: 908: 903: 898: 893: 888: 883: 878: 873: 867: 865: 861: 860: 858: 857: 847: 846: 841: 836: 826: 825: 820: 815: 810: 805: 795: 794: 789: 784: 779: 774: 769: 764: 759: 754: 749: 743: 738: 733: 728: 723: 718: 713: 708: 703: 698: 693: 688: 683: 678: 673: 668: 663: 658: 653: 648: 643: 638: 633: 628: 623: 618: 613: 608: 596: 594: 587: 581: 580: 571: 569: 568: 561: 554: 546: 539: 538: 495: 446: 413:Sci Transl Med 402: 350: 314: 285: 266: 264: 261: 248:. It binds to 233: 232: 222: 216: 215: 212: 206: 200: 194: 188: 183: 177: 176: 172: 171: 169: 168: 160: 158: 152: 151: 149: 148: 140: 138: 132: 131: 129: 128: 124: 122: 116: 115: 113: 112: 104: 102: 96: 95: 91: 90: 88: 87: 83: 81: 75: 74: 70: 69: 64: 58: 57: 47: 41: 40: 39:Whole antibody 37: 31: 30: 15: 13: 10: 9: 6: 4: 3: 2: 1706: 1695: 1692: 1690: 1687: 1685: 1682: 1680: 1677: 1675: 1672: 1671: 1669: 1658: 1653: 1651: 1646: 1644: 1639: 1638: 1632: 1630: 1626: 1622: 1617: 1614: 1610: 1593: 1591: 1588: 1587: 1585: 1582: 1579: 1576: 1574: 1571: 1570: 1566: 1556: 1553: 1551: 1548: 1546: 1543: 1541: 1538: 1537: 1535: 1531: 1528: 1526: 1523:Inflammatory 1521: 1511: 1508: 1507: 1505: 1501: 1495: 1494:Tildrakizumab 1492: 1490: 1487: 1485: 1482: 1480: 1477: 1475: 1472: 1470: 1467: 1465: 1462: 1460: 1457: 1455: 1452: 1450: 1447: 1445: 1442: 1440: 1437: 1436: 1434: 1430: 1424: 1421: 1419: 1416: 1414: 1411: 1409: 1406: 1404: 1401: 1399: 1396: 1394: 1391: 1389: 1386: 1384: 1381: 1379: 1376: 1374: 1371: 1370: 1368: 1364: 1361: 1359: 1355: 1345: 1342: 1340: 1337: 1335: 1332: 1331: 1329: 1324: 1320: 1319: 1316: 1312: 1308: 1301: 1298: 1296: 1295:Vobarilizumab 1293: 1291: 1288: 1286: 1283: 1281: 1278: 1276: 1273: 1271: 1268: 1266: 1263: 1261: 1258: 1256: 1253: 1251: 1248: 1246: 1243: 1241: 1240:Spartalizumab 1238: 1236: 1233: 1231: 1228: 1226: 1223: 1221: 1218: 1216: 1213: 1211: 1208: 1206: 1203: 1201: 1198: 1196: 1193: 1191: 1188: 1186: 1183: 1181: 1178: 1176: 1173: 1171: 1168: 1166: 1165:Pembrolizumab 1163: 1161: 1158: 1156: 1153: 1151: 1148: 1146: 1143: 1140: 1136: 1133: 1131: 1128: 1126: 1125:Mogamulizumab 1123: 1121: 1118: 1116: 1113: 1111: 1108: 1106: 1103: 1101: 1098: 1096: 1093: 1091: 1088: 1086: 1083: 1081: 1078: 1076: 1073: 1071: 1068: 1066: 1063: 1061: 1058: 1056: 1053: 1051: 1048: 1046: 1045:Crizanlizumab 1043: 1041: 1038: 1036: 1033: 1031: 1028: 1026: 1023: 1021: 1018: 1016: 1013: 1011: 1008: 1005: 1004: 1002: 1000: 996: 990: 987: 985: 982: 980: 977: 975: 972: 970: 967: 965: 962: 960: 957: 955: 952: 950: 947: 945: 942: 940: 939:Andecaliximab 937: 936: 934: 932: 928: 922: 919: 917: 914: 912: 909: 907: 904: 902: 899: 897: 894: 892: 889: 887: 884: 882: 879: 877: 874: 872: 869: 868: 866: 862: 856: 852: 849: 848: 845: 842: 840: 837: 835: 831: 828: 827: 824: 821: 819: 816: 814: 811: 809: 806: 804: 800: 797: 796: 793: 790: 788: 785: 783: 780: 778: 775: 773: 770: 768: 765: 763: 760: 758: 755: 753: 750: 747: 744: 742: 739: 737: 734: 732: 729: 727: 724: 722: 719: 717: 714: 712: 709: 707: 704: 702: 699: 697: 694: 692: 689: 687: 684: 682: 679: 677: 674: 672: 669: 667: 664: 662: 659: 657: 654: 652: 649: 647: 644: 642: 639: 637: 634: 632: 629: 627: 624: 622: 619: 617: 614: 612: 609: 607: 603: 602: 598: 597: 595: 591: 588: 586: 585:Immune system 582: 578: 577:immune system 574: 567: 562: 560: 555: 553: 548: 547: 544: 534: 530: 526: 522: 518: 514: 510: 506: 499: 496: 491: 487: 482: 477: 473: 469: 465: 461: 457: 450: 447: 442: 438: 434: 430: 426: 422: 418: 414: 406: 403: 398: 394: 389: 384: 379: 374: 370: 366: 362: 354: 351: 346: 342: 338: 334: 330: 326: 318: 315: 310: 306: 299: 295: 289: 286: 282: 281: 276: 271: 268: 262: 260: 258: 253: 251: 247: 243: 239: 223: 221: 217: 184: 182: 178: 173: 166: 162: 161: 159: 157: 153: 146: 142: 141: 139: 137: 133: 126: 125: 123: 121: 117: 110: 106: 105: 103: 101: 97: 92: 85: 84: 82: 80: 76: 73:Clinical data 71: 68: 65: 63: 59: 55: 51: 48: 46: 42: 38: 36: 32: 29: 25: 1629:expanding it 1618: 1484:Risankizumab 1469:Lebrikizumab 1449:Clazakizumab 1439:Anrukinzumab 1418:Tralokinumab 1334:Otelixizumab 1314: 1306: 1305: 1275:Tregalizumab 1260:Tislelizumab 1230:Satralizumab 1210:Rontalizumab 1205:Retifanlimab 1189: 1180:Plozalizumab 1160:Pateclizumab 1155:Pascolizumab 1150:Ozoralizumab 1100:Lampalizumab 1090:Inebilizumab 1080:Fontolizumab 1030:Camrelizumab 1025:Benralizumab 1020:Atezolizumab 1006: 949:Clenoliximab 850: 834:Bertilimumab 829: 818:Tremelimumab 798: 721:Mavrilimumab 711:Lirentelimab 706:Lerdelimumab 681:Fresolimumab 621:Atorolimumab 599: 508: 504: 498: 466:(1): 22–29. 463: 459: 449: 416: 412: 405: 368: 364: 353: 328: 324: 317: 308: 304: 288: 278: 270: 254: 237: 236: 109:1228538-47-3 1580:from market 1550:Lemalesomab 1545:Fanolesomab 1540:Besilesomab 1479:Perakizumab 1464:Mirikizumab 1454:Gevokizumab 1444:Bimekizumab 1423:Ustekinumab 1408:Secukinumab 1393:Fezakinumab 1388:Canakinumab 1383:Briakinumab 1358:Interleukin 1311:Dostarlimab 1290:Visilizumab 1285:Vedolizumab 1280:Vatelizumab 1270:Toralizumab 1265:Tocilizumab 1250:Teclistamab 1225:Samalizumab 1215:Rovelizumab 1195:Ravulizumab 1175:Pidilizumab 1170:Pexelizumab 1135:Ocrelizumab 1130:Natalizumab 1120:Mepolizumab 1110:Ligelizumab 1105:Letolizumab 1075:Etrolizumab 1065:Epratuzumab 1035:Cedelizumab 989:Vapaliximab 984:Teneliximab 974:Lumiliximab 959:Gomiliximab 944:Basiliximab 916:Vepalimomab 901:Nerelimomab 886:Gavilimomab 881:Faralimomab 876:Elsilimomab 851:Combination 844:Zanolimumab 839:Ontamalimab 787:Ulocuplumab 782:Tezepelumab 772:Sifalimumab 752:Pamrevlumab 731:Morolimumab 726:Metelimumab 696:Lanadelumab 631:Avdoralimab 616:Anifrolumab 365:Respir. Res 231: g·mol 94:Identifiers 1668:Categories 1510:Lokivetmab 1503:Veterinary 1489:Spesolimab 1474:Olokizumab 1459:Ixekizumab 1403:Guselkumab 1398:Fletikumab 1378:Brazikumab 1373:Bermekimab 1344:Sutimlimab 1318:Ibalizumab 1255:Teplizumab 1235:Siplizumab 1220:Ruplizumab 1200:Reslizumab 1190:Quilizumab 1145:Omalizumab 1095:Itolizumab 1085:Frexalimab 1060:Efalizumab 1055:Eculizumab 1050:Daclizumab 1015:Aselizumab 1010:Apolizumab 979:Priliximab 964:Infliximab 906:Odulimomab 896:Maslimomab 891:Inolimomab 871:Afelimomab 808:Durvalumab 803:Ipilimumab 792:Varlilumab 762:Relatlimab 757:Placulumab 701:Lenzilumab 676:Emapalumab 661:Cemiplimab 646:Brodalumab 641:Bleselumab 611:Adalimumab 263:References 238:Quilizumab 220:Molar mass 145:26F96HRJ3W 120:ChemSpider 100:CAS Number 21:Quilizumab 1590:Phase III 1578:Withdrawn 1555:Sulesomab 1432:Humanized 1413:Sirukumab 1245:Talizumab 1070:Erlizumab 999:Humanized 969:Keliximab 954:Galiximab 813:Nivolumab 777:Tabalumab 767:Sarilumab 741:Oleclumab 736:Namilumab 716:Lirilumab 691:Ianalumab 686:Golimumab 671:Eldelumab 666:Dupilumab 636:Belimumab 606:Abrilumab 257:Genentech 50:Humanized 931:Chimeric 823:Urelumab 746:Oxelumab 656:Carlumab 626:Avelumab 575:for the 533:51710078 525:30033912 490:29290750 441:41593528 433:24990880 397:26993628 345:27567329 296:(2011). 79:ATC code 1525:lesions 1300:TGN1412 1185:PRO 140 481:5735517 388:4797126 181:Formula 1573:WHO-EM 1315:Other: 531:  523:  488:  478:  439:  431:  395:  385:  371:: 29. 343:  246:asthma 165:D10409 62:Target 52:(from 45:Source 1619:This 1533:Mouse 1366:Human 864:Mouse 830:Other 593:Human 529:S2CID 437:S2CID 301:(PDF) 195:10046 54:mouse 1625:stub 521:PMID 486:PMID 429:PMID 393:PMID 341:PMID 311:(4). 250:IGHE 207:2023 201:1728 189:6492 156:KEGG 136:UNII 127:none 86:none 67:IGHE 35:Type 513:doi 476:PMC 468:doi 421:doi 383:PMC 373:doi 333:doi 329:138 242:INN 229:.49 227:082 225:146 1670:: 1586:: 1309:: 853:: 832:: 801:: 604:: 527:. 519:. 507:. 484:. 474:. 464:13 462:. 458:. 435:. 427:. 415:. 391:. 381:. 369:17 367:. 363:. 339:. 327:. 309:25 307:. 303:. 277:, 259:. 252:. 213:44 1656:e 1649:t 1642:v 1631:. 1141:) 1137:( 748:§ 565:e 558:t 551:v 535:. 515:: 509:6 492:. 470:: 443:. 423:: 417:6 399:. 375:: 347:. 335:: 283:. 240:( 210:S 204:O 198:N 192:H 186:C 56:)

Index

Monoclonal antibody
Type
Source
Humanized
mouse
Target
IGHE
ATC code
CAS Number
1228538-47-3
ChemSpider
UNII
26F96HRJ3W
KEGG
D10409
Formula
Molar mass
INN
asthma
IGHE
Genentech
Statement On A Nonproprietary Name Adopted By The USAN Council - Quilizumab
American Medical Association
World Health Organization
"International Nonproprietary Names for Pharmaceutical Substances (INN). Proposed INN: List 106"
doi
10.1016/j.jaci.2016.06.023
PMID
27567329
"A randomized trial of the efficacy and safety of quilizumab in adults with inadequately controlled allergic asthma"

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